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In vivo characterization of novel full and partial 2-(4-aminophenyl)-N,N-dipropylethylamine dopamine D2 receptor agonists

✍ Scribed by Sven Ahlenius; EvaLena Ericson; Lennart Florvall; Patricia Jiménez; Viveka Hillegaart; Agneta Wijkström


Book ID
114012932
Publisher
Elsevier Science
Year
2000
Tongue
English
Weight
259 KB
Volume
394
Category
Article
ISSN
0014-2999

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The present study was designed to characterize the dopamine D 3 receptor agonist R()-7-hydroxy-N,N-di-n-propyl-2-aminotetralin (R()-7-OH-DPAT)-induced changes in locomotor activity in mice. Although R()-7-OH-DPAT (0 . 01±10 mg/kg) produced a signi®cant decrease in horizontal and vertical motility wi