Hydroxymethylation and aminomethylation of 2-imino-5-arylidenethiazolidin-4-ones
✍ Scribed by S. Yu. Solov'eva-Yavits; S. M. Ramsh; N. A. Smorygo; A. I. Ginak; E. G. Sochilin
- Book ID
- 112370062
- Publisher
- Springer US
- Year
- 1980
- Tongue
- English
- Weight
- 306 KB
- Volume
- 16
- Category
- Article
- ISSN
- 0009-3122
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## Abstract New 2‐(aminomethyl)‐5‐(hydroxymethyl)pyrrolidine‐3,4‐diol derivatives were synthesized from (5__S__)‐5‐[(trityloxy)methyl]pyrrolidin‐2‐one (**6**) (__Schemes 1__ and __2__) and their inhibitory activities toward 25 glycosidases assayed (__Table__). The influence of the configuration of
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