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High-affinity fluorescent ligands for the 5-HT3 receptor

✍ Scribed by Jonathan Simonin; Sanjeev Kumar V. Vernekar; Andrew J. Thompson; J. Daniel Hothersall; Christopher N. Connolly; Sarah C.R. Lummis; Martin Lochner

Book ID
113496430
Publisher
Elsevier Science
Year
2012
Tongue
English
Weight
504 KB
Volume
22
Category
Article
ISSN
0960-894X

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Hindered rotation congeners of mazaperti
Hindered rotation congeners of mazapertine: High affinity ligands for the 5-HT1A receptor
✍ Ellen W. Baxter; Allen B. Reitz πŸ“‚ Article πŸ“… 1997 πŸ› Elsevier Science 🌐 English βš– 293 KB

Hindered rotation analogs of the antipsychotic mazapertine (1) were prepared. These compounds exhibited high affinity for the 5-HTl\* receptor, but not for other serotonin or dopamine receptors. The related p carboline structures were also synthesized and were found to he potent .S-HT~A ligands. 0 1