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Flecainide enantiomers: Disposition in human subjects and electrophysiologic actions in vitro

✍ Scribed by Kroemer, Heyo K; Turgeon, Jacques; Parker, Robert A; Roden, Dan M


Book ID
109844607
Publisher
Nature Publishing Group
Year
1989
Tongue
English
Weight
516 KB
Volume
46
Category
Article
ISSN
0009-9236

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## Abstract Pharmacokinetics of sulpiride enantiomers after intravenous administration of (Β±)‐, (+)‐, and (βˆ’)‐sulpiride was examined in humans and rats. Pharmacokinetic profiles were similar in (+)‐ and (βˆ’)‐enantiomers after intravenous administration of (Β±)‐sulpiride. Metabolic inversion at a chir