A new series of DNA binding 5,10,15-tri(N-methyl-4-pyridiniumyl)porphyrin (TrisMPyP)-platinum(II) conjugates was synthesized, in which different spacer ligands were used for appropriate coordination to platinum(II) complexes. Compound 9b exhibited in vivo antitumor activity (T/C%, 294) superior to c
β¦ LIBER β¦
DNA-binding properties of antitumor-activecis-bis(pyridine)platinum(II) organoamides
β Scribed by Marieke J. Bloemink; Robert J. Heetebrij; Joanne Ireland; Glen B. Deacon; J. Reedijk
- Publisher
- John Wiley and Sons
- Year
- 1996
- Tongue
- English
- Weight
- 188 KB
- Volume
- 1
- Category
- Article
- ISSN
- 1432-1327
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