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Discovery of (( S )-5-(Methoxymethyl)-7-(1-methyl-1 H -indol-2-yl)-2-(trifluoromethyl)-4,7-dihydropyrazolo[1,5- a ]pyrimidin-6-yl)(( S )-2-(3-methylisoxazol-5-yl)pyrrolidin-1-yl)methanone As a Potent and Selective I Kur Inhibitor

✍ Scribed by Finlay, Heather J.; Lloyd, John; Vaccaro, Wayne; Kover, Alexander; Yan, Lin; Bhave, Gauri; Prol, Joseph; Huynh, Tram; Bhandaru, Rao; Caringal, Yolanda; DiMarco, John; Gan, Jinping; Harper, Tim; Huang, Christine; Conder, Mary Lee; Sun, Huabin; Levesque, Paul; Blanar, Michael; Atwal, Karnail; Wexler, Ruth

Book ID: 118036686
Publisher: American Chemical Society
Year: 2012
Tongue: English
Weight: 465 KB
Volume: 55
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm201386u

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