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Discovery of pyrazolo[1,5-a]pyrimidine-based Pim inhibitors: A template-based approach

✍ Scribed by Dwyer, Michael P.; Keertikar, Kartik; Paruch, Kamil; Alvarez, Carmen; Labroli, Marc; Poker, Cory; Fischmann, Thierry O.; Mayer-Ezell, Rosemary; Bond, Richard; Wang, Yan; Azevedo, Rita; Guzi, Timothy J.


Book ID
121190670
Publisher
Elsevier Science
Year
2013
Tongue
English
Weight
616 KB
Volume
23
Category
Article
ISSN
0960-894X

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## Abstract Naphtho[2,1‐__b__]furan‐2‐yl)(8‐phenylpyrazolo[5,1‐__c__][1,2,4]triazin‐3‐yl)methanone, ([1,2,4]triazolo[3,4‐__c__][1,2,4]triazin‐6‐yl)(naphtho[2,1‐__b__]furan‐2‐yl)methanone, benzo[4,5]imidazo[2,1‐__c__][1,2,4]triazin‐3‐yl‐naphtho[2,1‐__b__]furan‐2‐yl‐methanone, 5‐(naphtho[2,1‐__b__]fu