Discovery of Diaryl Imidazolidin-2-one Derivatives, a Novel Class of Muscarinic M3 Selective Antagonists (Part 1)
✍ Scribed by Peretto, Ilaria; Forlani, Roberto; Fossati, Claudia; Giardina, Giuseppe A. M.; Giardini, Alessandra; Guala, Matilde; La Porta, Elena; Petrillo, Paola; Radaelli, Stefano; Radice, Luigi; Raveglia, Luca F.; Santoro, Enza; Scudellaro, Roberta; Scarpitta, Francesca; Bigogno, Chiara; Misiano, Paola; Dondio, Giulio M.; Rizzi, Andrea; Armani, Elisabetta; Amari, Gabriele; Civelli, Maurizio; Villetti, Gino; Patacchini, Riccardo; Bergamaschi, Marco; Delcanale, Maurizio; Salcedo, Carolina; Fernández, Andrés G.; Imbimbo, Bruno P.
- Book ID
- 126881057
- Publisher
- American Chemical Society
- Year
- 2007
- Tongue
- English
- Weight
- 436 KB
- Volume
- 50
- Category
- Article
- ISSN
- 0022-2623
No coin nor oath required. For personal study only.
📜 SIMILAR VOLUMES
Synthesis of Novel Succinamide Derivatives Having a 5,11-Dihydro-6H-pyrido[2,3-b][1,4]benzodiazepin-6-one Skeleton as Potent and Selective M 2 Muscarinic Receptor Antagonists. Part 2. -Among the screened compounds derivative (IIIe) exhibits the highest affinity for M 2 muscarinic receptors and (III