✦ LIBER ✦

Discovery of Dermorphin-Based Affinity Labels with Subnanomolar Affinity for Mu Opioid Receptors †

✍ Scribed by Sinha, Bhaswati; Cao, Zhengyu; Murray, Thomas F.; Aldrich, Jane V.

Book ID: 119998682
Publisher: American Chemical Society
Year: 2009
Tongue: English
Weight: 708 KB
Volume: 52
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm9007592

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Affinity labelling of mu opioid receptor

Affinity labelling of mu opioid receptors

✍ A. Borsodi; H.A. Öktem; S. Benyhe; É. Varga; J. Moitra; J. Takács; A. Lajtha 📂 Article 📅 1990 🏛 Elsevier Science 🌐 English ⚖ 227 KB

Synthesis of enkephalin-based affinity l

Synthesis of enkephalin-based affinity labels for delta opioid receptors

✍ DY Maeda; TF Murray; JE Roth; JV Aldrich 📂 Article 📅 1994 🏛 Elsevier Science 🌐 English ⚖ 114 KB

32P Labeled Opioid Peptides with High Af

32P Labeled Opioid Peptides with High Affinity for the δ-Opioid Receptor

✍ B.L. Kieffer; D. Black; C.G. Hirth 📂 Article 📅 1993 🏛 Elsevier Science 🌐 English ⚖ 748 KB

Tyr-D-Ala-Gly-(Me)Phe-chloromethyl keton

Tyr-D-Ala-Gly-(Me)Phe-chloromethyl ketone: A mu specific affinity label for the opioid receptor

✍ S Benyhe; J Hepp; J Simon; A Borsodi; K Medzihradszky; M Wollemann 📂 Article 📅 1987 🏛 Elsevier Science 🌐 English ⚖ 700 KB

Affinity labels as tools for the identif

Affinity labels as tools for the identification of opioid receptor recognition sites

✍ Philip S Portoghese; Rachid El Kouhen; Ping Y Law; Horace H Loh; Bertrand Le Bou 📂 Article 📅 2001 🏛 Elsevier Science 🌐 English ⚖ 165 KB

Synthesis and evaluation of derivatives

Synthesis and evaluation of derivatives of leucine enkephalin as potential affinity labels for δ opioid receptors

✍ Heekyung Choi; Thomas F. Murray; Jane V. Aldrich 📂 Article 📅 2003 🏛 Wiley (John Wiley & Sons) 🌐 English ⚖ 82 KB

As part of an effort to develop peptide-based affinity labels for opioid receptors, [Leu(5)]enkephalin (LeuEnk) and DTLET (Tyr-D-Thr-Gly-Phe-Leu-Thr), potent agonists for delta receptors, were selected as the parent peptides for further modification. The affinity label derivatives were prepared usin