Discovery of a Selective, Substrate-Competitive Inhibitor of the Lysine Methyltransferase SETD8

✍ Scribed by Ma, Anqi; Yu, Wenyu; Li, Fengling; Bleich, Rachel M.; Herold, J. Martin; Butler, Kyle V.; Norris, Jacqueline L.; Korboukh, Victoria; Tripathy, Ashutosh; Janzen, William P.; Arrowsmith, Cheryl H.; Frye, Stephen V.; Vedadi, Masoud; Brown, Peter J.; Jin, Jian

• Book ID: 127013059
• Publisher: American Chemical Society
• Year: 2014
• Tongue: English
• Weight: 1024 KB
• Volume: 57
• Category: Article
• ISSN: 0022-2623
• DOI: 10.1021/jm500871s