✦ LIBER ✦

Discovery of a subtype selective inhibitor of the human betaine/GABA transporter 1 (BGT-1) with a non-competitive pharmacological profile

✍ Scribed by Kragholm, Bolette; Kvist, Trine; Madsen, Karsten K.; Jørgensen, Lars; Vogensen, Stine B.; Schousboe, Arne; Clausen, Rasmus P.; Jensen, Anders A.; Bräuner-Osborne, Hans

Book ID: 122625986
Publisher: Elsevier Science
Year: 2013
Tongue: English
Weight: 549 KB
Volume: 86
Category: Article
ISSN: 0006-2952
DOI: 10.1016/j.bcp.2013.06.007

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Pharmacological Identification of a Guan

Pharmacological Identification of a Guanidine-Containing β-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

✍ Al-Khawaja, Anas; Petersen, Jette G.; Damgaard, Maria; Jensen, Mette H.; Vogense 📂 Article 📅 2014 🏛 Springer 🌐 English ⚖ 446 KB

Discovery of the First Selective Inhibit

Discovery of the First Selective Inhibitor of Excitatory Amino Acid Transporter Subtype 1

✍ Jensen, Anders A.; Erichsen, Mette N.; Nielsen, Christina W.; Stensbøl, Tine B.; 📂 Article 📅 2009 🏛 American Chemical Society 🌐 English ⚖ 136 KB

1-(3-(9H-Carbazol-9-yl)-1-propyl)-4-(2-m

1-(3-(9H-Carbazol-9-yl)-1-propyl)-4-(2-methoxyphenyl)-4-piperidinol, a novel subtype selective inhibitor of the mouse type II GABA-transporter

✍ Christian Thomsen; Per Olaf Sørensen; Jan Egebjerg 📂 Article 📅 1997 🏛 Nature Publishing Group 🌐 English ⚖ 382 KB

A single amino acid of the human and rat

A single amino acid of the human and rat neurotensin receptors (subtype 1) determining the pharmacological profile of a species-selective neurotensin agonist

✍ Bernadette Cusack; Karen Jansen; Daniel J McCormick; Thomas Chou; Yuan-Ping Pang 📂 Article 📅 2000 🏛 Elsevier Science 🌐 English ⚖ 404 KB

Discovery of GS-8374, a potent human imm

Discovery of GS-8374, a potent human immunodeficiency virus type 1 protease inhibitor with a superior resistance profile

✍ He, Gong-Xing; Yang, Zheng-Yu; Williams, Matthew; Callebaut, Christian; Cihlar, 📂 Article 📅 2011 🏛 The Royal Society of Chemistry 🌐 English ⚖ 209 KB

Gambogic Acid as a Non-Competitive Inhib

Gambogic Acid as a Non-Competitive Inhibitor of ATP-Binding Cassette Transporter B1 Reverses the Multidrug Resistance of Human Epithelial Cancers by Promoting ATP-Binding Cassette Transporter B1 Protein Degradation

✍ Xu Wang; Rongxin Deng; Yan Lu; Qin Xu; Ming Yan; Dongxia Ye; Wantao Chen 📂 Article 📅 2012 🏛 John Wiley and Sons 🌐 English ⚖ 611 KB