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Discovery of a Novel, Selective, and Orally Bioavailable Class of Thrombin Inhibitors Incorporating Aminopyridyl Moieties at the P1 Position

✍ Scribed by Feng, Dong-Mei; Gardell, Stephen J.; Lewis, S. Dale; Bock, Mark G.; Chen, Zhongguo; Freidinger, Roger M.; Naylor-Olsen, Adel M.; Ramjit, Harri G.; Woltmann, Richard; Baskin, Elizabeth P.; Lynch, Joseph J.; Lucas, Robert; Shafer, Jules A.; Dancheck, Kimberley B.; Chen, I-Wu; Mao, Shi-Shan; Krueger, Julie A.; Hare, Timothy R.; Mulichak, Anne M.; Vacca, Joseph P.

Book ID: 121482153
Publisher: American Chemical Society
Year: 1997
Tongue: English
Weight: 241 KB
Volume: 40
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm970493r

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