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Discovery of 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-7-(2,2-difluoropropyl)-6,7-dihydro-2 H -pyrazolo[3,4- f ][1,4]oxazepin-8(5 H )-one (PF-514273), a Novel, Bicyclic Lactam-Based Cannabinoid-1 Receptor Antagonist for the Treatment of Obesity

✍ Scribed by Dow, Robert L.; Carpino, Philip A.; Hadcock, John R.; Black, Shawn C.; Iredale, Philip A.; DaSilva-Jardine, Paul; Schneider, Steven R.; Paight, Ernest S.; Griffith, David A.; Scott, Dennis O.; O’Connor, Rebecca E.; Nduaka, Chudy I.

Book ID: 120629685
Publisher: American Chemical Society
Year: 2009
Tongue: English
Weight: 191 KB
Volume: 52
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm900255t

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