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Discovery of 1-[3-(Aminomethyl)phenyl]-N-[3-fluoro-2‘-(methylsulfonyl)- [1,1‘-biphenyl]-4-yl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide (DPC423), a Highly Potent, Selective, and Orally Bioavailable Inhibitor of Blood Coagulation Factor Xa1

✍ Scribed by Pinto, Donald J. P.; Orwat, Michael J.; Wang, Shuaige; Fevig, John M.; Quan, Mimi L.; Amparo, Eugene; Cacciola, Joseph; Rossi, Karen A.; Alexander, Richard S.; Smallwood, Angela M.

Book ID: 115476535
Publisher: American Chemical Society
Year: 2001
Tongue: English
Weight: 320 KB
Volume: 44
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm000409z

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