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Discovery of 1-(2-Aminomethylphenyl)-3-trifluoromethyl- N - [3-fluoro-2‘-(aminosulfonyl)[1,1‘-biphenyl)]-4-yl]-1 H -pyrazole-5-carboxyamide (DPC602), a Potent, Selective, and Orally Bioavailable Factor Xa Inhibitor 1

✍ Scribed by Pruitt, James R.; Pinto, Donald J. P.; Galemmo,, Robert A.; Alexander, Richard S.; Rossi, Karen A.; Wells, Brian L.; Drummond, Spencer; Bostrom, Lori L.; Burdick, Debra; Bruckner, Robert; Chen, Haiying; Smallwood, Angela; Wong, Pancras C.; Wright, Matthew R.; Bai, Steven; Luettgen, Joseph M.; Knabb, Robert M.; Lam, Patrick Y. S.; Wexler, Ruth R.

Book ID: 120052135
Publisher: American Chemical Society
Year: 2003
Tongue: English
Weight: 555 KB
Volume: 46
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm030212h

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