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Discovery and Characterization of 6-{4-[3-( R )-2-Methylpyrrolidin-1-yl)propoxy]phenyl}-2 H -pyridazin-3-one (CEP-26401, Irdabisant): A Potent, Selective Histamine H 3 Receptor Inverse Agonist

✍ Scribed by Hudkins, Robert L.; Raddatz, Rita; Tao, Ming; Mathiasen, Joanne R.; Aimone, Lisa D.; Becknell, Nadine C.; Prouty, Catherine P.; Knutsen, Lars J. S.; Yazdanian, Mehran; Moachon, Gilbert; Ator, Mark A.; Mallamo, John P.; Marino, Michael J.; Bacon, Edward R.; Williams, Michael

Book ID: 118260263
Publisher: American Chemical Society
Year: 2011
Tongue: English
Weight: 1007 KB
Volume: 54
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm200401v

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