Inhibitory activity and selectivity of s
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Giorgio Caravatti; Thomas Meyer; Andreas Fredenhagen; Uwe Trinks; Helmut Mett; D
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Article
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1994
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Elsevier Science
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English
β 440 KB
Abbractz The synthesis sod b vibu protein kinase C (PKC) inhibition ofa series of staurosporine derivatives is descrii. Essential foractivityisafneNHofIhcLadampwtionofthemolecule.Alargevarictyofarbslitucntsistolcra~atthcsecondaryamine, altlwugh in mcst cases these modifications I& to a dccrrasc in a