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Development of Human Calcitonin Gene-Related Peptide (CGRP) Receptor Antagonists. 1. Potent and Selective Small Molecule CGRP Antagonists. 1-[ N 2 -[3,5-Dibromo- N -[[4-(3,4-dihydro-2(1 H )-oxoquinazolin-3-yl)-1- piperidinyl]carbonyl]- d -tyrosyl]- l -lysyl]-4-(4-pyridinyl)piperazine: The First CGRP Antagonist for Clinical Trials in Acute Migraine †

✍ Scribed by Rudolf, Klaus; Eberlein, Wolfgang; Engel, Wolfhard; Pieper, Helmut; Entzeroth, Michael; Hallermayer, Gerhard; Doods, Henri

Book ID
120379645
Publisher
American Chemical Society
Year
2005
Tongue
English
Weight
222 KB
Volume
48
Category
Article
ISSN
0022-2623

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