## Abstract The in silico design, synthesis, and biological evaluation of ten potent type II dehydroquinase inhibitors are described. These compounds contain an anhydroquinate core, incorporated as a mimic of the enolate reaction intermediate. This substructure is attached by a variety of linking u
✦ LIBER ✦
Design, Synthesis, and Structural Studies on Potent Biaryl Inhibitors of Type II Dehydroquinases
✍ Scribed by Richard J. Payne; Alan Riboldi-Tunnicliffe; Olivier Kerbarh; Andrew D. Abell; Adrian J. Lapthorn; Chris Abell
- Publisher
- John Wiley and Sons
- Year
- 2007
- Tongue
- English
- Weight
- 286 KB
- Volume
- 2
- Category
- Article
- ISSN
- 1860-7179
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