✦ LIBER ✦

Derivatives of the Triazoloquinazoline Adenosine Antagonist (CGS15943) Are Selective for the Human A3 Receptor Subtype

✍ Scribed by Kim, Yong-Chul; Ji, Xiao-duo; Jacobson, Kenneth A.

Book ID: 111867749
Publisher: American Chemical Society
Year: 1996
Tongue: English
Weight: 289 KB
Volume: 39
Category: Article
ISSN: 0022-2623
DOI: 10.1021/jm960482i

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

ChemInform Abstract: Derivatives of the

ChemInform Abstract: Derivatives of the Triazoloquinazoline Adenosine Antagonist (CGS15943) (I) are Selective for the Human A3 Receptor Subtype.

✍ Y.-C. KIM; X. JI; K. A. JACOBSON 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 30 KB 👁 1 views

Derivatives of the Triazoloquinazoline A

Derivatives of the Triazoloquinazoline Adenosine Antagonist (CGS 15943) Having High Potency at the Human A 2B and A 3 Receptor Subtypes

✍ Kim, Yong-Chul; de Zwart, Maarten; Chang, Louis; Moro, Stefano; von Frijtag Drab 📂 Article 📅 1998 🏛 American Chemical Society 🌐 English ⚖ 202 KB

Comparison of the behavioural effects of

Comparison of the behavioural effects of an adenosine A1/A2-receptor antagonist, CGS 15943A, and an A1-selective antagonist, DPCPX

✍ Guy Griebel; Martine Saffroy-Spittler; René Misslin; Delphine Remmy; Elise Vogel 📂 Article 📅 1991 🏛 Springer 🌐 English ⚖ 563 KB

QSAR of adenosine receptor antagonists.

QSAR of adenosine receptor antagonists. Part 3: Exploring physicochemical requirements for selective binding of 1,2,4-triazolo[5,1-i]purine derivatives with human adenosine A3 receptor subtype

✍ Kunal Roy; J.Thomas Leonard; Chandana Sengupta 📂 Article 📅 2004 🏛 Elsevier Science 🌐 English ⚖ 257 KB

Potent antagonists for the human adenosi

Potent antagonists for the human adenosine A2B receptor. Derivatives of the triazolotriazine adenosine receptor antagonist ZM241385 with high affinity

✍ Maarten de Zwart; Roel C. Vollinga; Margot W. Beukers; Danielle F. Sleegers; Jac 📂 Article 📅 1999 🏛 John Wiley and Sons 🌐 English ⚖ 147 KB 👁 2 views

A series of novel and known 5-substituted 7-amino-2-(2-furyl) [1,2,4]triazolo [1,5a][1,3,5]triazine derivatives were synthesized and tested for adenosine receptor antagonism in radioligand binding assays at all four adenosine receptor subtypes and for inhibition of the agonist-induced cyclic AMP res

Generation of adenosine A3 receptor func

Generation of adenosine A3 receptor functionally humanized mice for the evaluation of the human antagonists

✍ Kazuya Yamano; Miho Inoue; Shigehiro Masaki; Mayumi Saki; Michio Ichimura; Mitsu 📂 Article 📅 2006 🏛 Elsevier Science 🌐 English ⚖ 639 KB