✦ LIBER ✦

Cyclic analogs of α-melanocyte-stimulating hormone (αMSH) with high agonist potency and selectivity at human melanocortin receptor 1b

✍ Scribed by Maria A. Bednarek; Tanya MacNeil; Rui Tang; Tung M. Fong; M. Angeles Cabello; Marta Maroto; Ana Teran

Book ID: 116831619
Publisher: Elsevier Science
Year: 2008
Tongue: English
Weight: 230 KB
Volume: 29
Category: Article
ISSN: 0196-9781
DOI: 10.1016/j.peptides.2008.02.008

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Analogs of α-melanocyte stimulating horm

Analogs of α-melanocyte stimulating hormone with high agonist potency and selectivity at human melanocortin receptor 1b: The role of Trp9 in molecular recognition

✍ Maria A. Bednarek; Tanya MacNeil; Rui Tang; Tung M. Fong; M. Angeles Cabello; Ma 📂 Article 📅 2008 🏛 Wiley (John Wiley & Sons) 🌐 English ⚖ 133 KB

## Abstract α‐Melanocyte stimulating hormone (αMSH), Ac‐Ser^1^‐Tyr^2^‐Ser^3^‐Met^4^‐Glu^5^‐His^6^‐Phe^7^‐Arg^8^‐Trp^9^‐Gly^10^‐Lys^11^‐Pro^12^‐Val^13^‐NH~2~, is an endogenous agonist for the melanocortin receptor 1 (MC1R), the receptor found in the skin, several types of immune cells, and other per

Potent and Selective Agonists of Human M

Potent and Selective Agonists of Human Melanocortin Receptor 5: Cyclic Analogues of α-Melanocyte-Stimulating Hormone †

✍ Bednarek, Maria A.; MacNeil, Tanya; Tang, Rui; Fong, Tung M.; Cabello, M. Angele 📂 Article 📅 2007 🏛 American Chemical Society 🌐 English ⚖ 66 KB

Potent and Selective Peptide Agonists of

Potent and Selective Peptide Agonists of α-Melanocyte Stimulating Hormone (αMSH) Action at Human Melanocortin Receptor 5; their Synthesis and Biological Evaluation in vitro

✍ Maria A. Bednarek; Tanya MacNeil; Rui Tang; Tung M. Fong; M. Angeles Cabello; Ma 📂 Article 📅 2007 🏛 John Wiley and Sons 🌐 English ⚖ 168 KB

Effects of Macrocycle Size and Rigidity

Effects of Macrocycle Size and Rigidity on Melanocortin Receptor-1 and -5 Selectivity in Cyclic Lactam α-Melanocyte-Stimulating Hormone Analogs

✍ Alexander V. Mayorov; So-Yeop Han; Minying Cai; Matthew R. Hammer; Dev Trivedi; 📂 Article 📅 2006 🏛 John Wiley and Sons 🌐 English ⚖ 113 KB

Potent and selective agonists of α-melan

Potent and selective agonists of α-melanotropin (αMSH) action at human melanocortin receptor 5; linear analogs of α-melanotropin

✍ Maria A. Bednarek; Tanya MacNeil; Rui Tang; Tung M. Fong; M. Angeles Cabello; Ma 📂 Article 📅 2007 🏛 Elsevier Science 🌐 English ⚖ 193 KB

Solid-phase peptide head-to-side chain c

Solid-phase peptide head-to-side chain cyclodimerization: Discovery of C2-symmetric cyclic lactam hybrid α-melanocyte-stimulating hormone (MSH)/agouti-signaling protein (ASIP) analogues with potent activities at the human melanocortin receptors

✍ Alexander V. Mayorov; Minying Cai; Erin S. Palmer; Zhihua Liu; James P. Cain; Jo 📂 Article 📅 2010 🏛 Elsevier Science 🌐 English ⚖ 625 KB