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Corrigendum to “Discovery of GSK1997132B a novel centrally penetrant benzimidazole PPARγ partial agonist” [Bioorg. Med. Chem. Lett. 21 (2011) 5568–5572]

✍ Scribed by Sime, Mairi; Allan, Amanda C.; Chapman, Paul; Fieldhouse, Charlotte; Giblin, Gerard M.P.; Healy, Mark P.; Lambert, Millard H.; Leesnitzer, Lisa M.; Lewis, Ann; Merrihew, Raymond V.; Rutter, Richard A.; Sasse, Rosemary; Shearer, Barry G.; Willson, Timothy M.; Xu, Robert X.; Virley, David J.

Book ID: 122981360
Publisher: Elsevier Science
Year: 2013
Tongue: English
Weight: 117 KB
Volume: 23
Category: Article
ISSN: 0960-894X
DOI: 10.1016/j.bmcl.2012.12.062

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ChemInform Abstract: Discovery of GSK199

ChemInform Abstract: Discovery of GSK1997132B a Novel Centrally Penetrant Benzimidazole PPARγ Partial Agonist.

✍ Mairi Sime; et al. et al. 📂 Article 📅 2011 🏛 John Wiley and Sons ⚖ 22 KB

## Abstract Optimization of the PPARγ activity and in vivo pharmacokinetics of a non‐acidic benzimidazole derivative, identified as starting point for a centrally penetrant PPARγ partial agonist, leads to the identification of title compound (I), a potent and metabolically stable PPARγ partial agon