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Copper-catalyzed cascade approach to 1,3-diazabicyclo[3.1.0]hex-3-enes from aziridines and ethyl diazoacetate

✍ Scribed by Yuanxun Zhu; Shaoyin Wang; Shan Wen; Ping Lu; Yanguang Wang

Publisher
Elsevier Science
Year
2010
Tongue
French
Weight
469 KB
Volume
51
Category
Article
ISSN
0040-4039

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✦ Synopsis

An efficient and general synthesis of 1,3-diazabicyclo[3.1.0]hex-3-enes via the copper-catalyzed cascade reaction of aziridines with ethyl diazoacetate is described.

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