The first synthesis of a combinatorial library using double combinatorial chemistry is presented. Coupling of unprotected Fmoc-tyrosine to the solid support was followed by Mitsunobu O-alkylation. Introduction of a diacid linker yields a system in which the double combinatorial step can be demonstra
β¦ LIBER β¦
Combinatorial synthesis of small-molecule libraries using 3-amino-5-hydroxybenzoic acid
β Scribed by Sharon M. Dankwardt; Thu M. Phan; John L. Krstenansky
- Book ID
- 105288493
- Publisher
- Springer
- Year
- 1996
- Tongue
- English
- Weight
- 641 KB
- Volume
- 1
- Category
- Article
- ISSN
- 1381-1991
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