The preparation of chiral pyrrolidine and piperidine b-enamino esters starting from v-halogeno b-keto esters, their diastereoselective reduction and the subsequent cleavage of the chiral auxiliary are described.
✦ LIBER ✦
Chiral Heterocyclic β-Enamino Esters: Convenient Synthesis and Diastereoselective Reduction.
✍ Scribed by Sandrine Calvet; Olivier David; Corinne Venucci-Bacque; Marie-Claude Fargeau-Bellassoued; Gerard Lhommet
- Publisher
- John Wiley and Sons
- Year
- 2003
- Weight
- 147 KB
- Volume
- 34
- Category
- Article
- ISSN
- 0931-7597
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