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Chemistry of acetylenic ethers XXXVII. Synthesis of β-lactams (2-azetidinones) from imines and ethoxyalkynes

✍ Scribed by A. M. van Leusen; J. F. Arens

Publisher
Elsevier Science
Year
2010
Tongue
English
Weight
346 KB
Volume
78
Category
Article
ISSN
0165-0513

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✦ Synopsis

Abstract

β‐Lactams VII are formed when ethoxyalkynes II are slowly added to boiling solutions of aromatic imines VI in xylene. In all probability aldoketenes III are intermediate products. The yields are moderate to good.

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