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ChemInform Abstract: Synthesis of Bis-heteroaryl Piperazine Derivatives as Potential Reverse Transcriptase Inhibitors.

โœ Scribed by Jean Guillaumel; David S. Grierson; Claude Monneret


Publisher
John Wiley and Sons
Year
2010
Weight
28 KB
Volume
32
Category
Article
ISSN
0931-7597

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ChemInform Abstract: Synthesis and Bioac
โœ M. J. GENIN; T. J. POEL; Y. YAGI; C. BILES; I. ALTHAUS; B. J. KEISER; L. A. KOPT ๐Ÿ“‚ Article ๐Ÿ“… 2010 ๐Ÿ› John Wiley and Sons โš– 33 KB ๐Ÿ‘ 2 views

Synthesis and Bioactivity of Novel Bis(heteroaryl)piperazine (BHAP) Reverse Transcriptase Inhibitors: Structure-Activity Relationships and Increased Metabolic Stability of Novel Substituted Pyridine Analogues. -Piperazine-containing compounds such as (VII) (11 examples) and piperidine containing an