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ChemInform Abstract: Synthesis of 14,17-Propano Analogues of Estradiol.

✍ Scribed by J. R. BULL; C. HOADLEY; P. G. MOUNTFORD; L. M. STEER

Publisher
John Wiley and Sons
Year
2010
Weight
31 KB
Volume
28
Category
Article
ISSN
0931-7597

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✦ Synopsis

Synthesis of 14,17-Propano Analogues of Estradiol.

-Novel interesting D-ring bridged estradiol derivatives such as (IV) and (VIII), which are further functionalized in the bridge, are synthesized. The results of the competitive binding assay toward the estradiol receptor are reported and discussed. -(BULL,

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