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ChemInform Abstract: Synthesis and Biological Evaluation of Dibenz[b,f][1,5]oxazocine Derivatives for Agonist Activity at ϰ-Opioid Receptor.

✍ Scribed by Sudipta Mitra; Tuhin Suvro Banerjee; Sandip K. Hota; Debleena Bhattacharya; Sumantra Das; Partha Chattopadhyay

Publisher: John Wiley and Sons
Year: 2011
Weight: 28 KB
Volume: 42
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.201131166

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✦ Synopsis

Abstract

A short synthetic route to title compounds (II) is developed using an optimized Pd‐catalyzed intramolecular cycloamination reaction as the key step.

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