ChemInform Abstract: Synthesis and Antifungal Properties of Benzylamines Containing Boronate Esters.
β Scribed by Christopher M. Vogels; Liliya G. Nikolcheva; David W. Norman; Heather A. Spinney; Andreas Decken; Mark O. Baerlocher; Felix J. Baerlocher; Stephen A. Westcott
- Publisher
- John Wiley and Sons
- Year
- 2010
- Weight
- 30 KB
- Volume
- 33
- Category
- Article
- ISSN
- 0931-7597
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Sulfonamides containing pinacol pro- tected boronate ester groups have been prepared by the addition of H 2 NC 6 H 4 Bpin (pin = O 2 C 2 Me 4 ) to sulfonyl chlorides p-RC 6 H 4 SO 2 Cl (R = CH 3 , NO 2 ). Hydrogenation of the nitro derivatives afford the corresponding sulfanilamides without compromi