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ChemInform Abstract: Ready Access to Enantiopure 5-Substituted-3-pyrrolin-2-ones from N-Benzyl-2,3-O-isopropylidene-D-glyceraldehyde Nitrone (BIGN).

✍ Scribed by P. MERINO; E. CASTILLO; S. FRANCO; F. L. MERCHAN; T. TEJERO

Publisher: John Wiley and Sons
Year: 2010
Weight: 35 KB
Volume: 29
Category: Article
ISSN: 0931-7597
DOI: 10.1002/chin.199841108

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✦ Synopsis

Ready Access to Enantiopure 5-Substituted-3-pyrrolin-2-ones from N-Benzyl-2,3-O-isopropylidene-D-glyceraldehyde Nitrone (BIGN).

-A short and efficient route to the title compounds is developed. These pyrrolinones are useful synthetic synthons and can be employed for the preparation of highly functionalized pyrrolidines.

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