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ChemInform Abstract: Copper-Catalyzed N-Arylation/Hydroamin(d)ation Domino Synthesis of Indoles and Its Application to the Preparation of a Chek1/KDR Kinase Inhibitor Pharmacophore.

✍ Scribed by Lutz Ackermann; Sebastian Barfuesser; Harish K. Potukuchi

Publisher
John Wiley and Sons
Year
2009
Weight
35 KB
Volume
40
Category
Article
ISSN
0931-7597

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Abstract

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Copper-Catalyzed N-Arylation/Hydroamin(d
Copper-Catalyzed N-Arylation/Hydroamin(d)ation Domino Synthesis of Indoles and its Application to the Preparation of a Chek1/KDR Kinase Inhibitor Pharmacophore
✍ Lutz Ackermann; Sebastian Barfüßer; Harish K. Potukuchi 📂 Article 📅 2009 🏛 John Wiley and Sons 🌐 English ⚖ 256 KB 👁 1 views

## Abstract magnified image Inexpensive copper catalysts allow for efficient syntheses of __N__‐aryl‐, __N__‐acyl‐, or __N__‐H‐(aza)indoles starting from __ortho__‐alkynylbromoarenes. The broad scope of this domino __N__‐arylation/hydroamin(d)ation process is highlighted by the synthesis of highly