Synthesis and 5Ξ±-Reductase Inhibitory Activities of Benzofuran Derivatives with a Carbamoyl Group. -5-Carbamoyl (VII) and 6-carbamoyl derivatives (XI) are prepared and found to show inhibitory activity of human 5Ξ±-reductase. The key step furan ring cyclization occurs by using HCl, cf. product (V),
ChemInform Abstract: Aminolysis of Methoxy Groups in Pyrimidine Derivatives. Activation by 5-Nitroso Group.
β Scribed by M. Melguizo; A. Marchal; M. Nogueras; A. Sanchez; J. N. Low
- Publisher
- John Wiley and Sons
- Year
- 2010
- Weight
- 29 KB
- Volume
- 33
- Category
- Article
- ISSN
- 0931-7597
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β¦ Synopsis
Abstract
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