Fluorescein-labeled stable neurotensin d
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Veronique Maes; Christina Hultsch; Suzann Kohl; Ralf Bergmann; Thomas Hanke; Dir
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Article
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2006
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John Wiley and Sons
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English
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Neurotensin(8-13) analogs containing a glycine or 5-aminovaleroyl spacer were labeled with fluorescein through formation of an N-terminal thiourea function. The receptor binding was measured in HT-29 cell cultures and showed a substantial decrease in affinity, especially for the metabolically stabil