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Aromatic Enamide/Ene Metathesis toward Substituted Indoles and Its Application to the Synthesis of Indomethacins

✍ Scribed by Yayoi Kasaya; Kosuke Hoshi; Yukiyoshi Terada; Atsushi Nishida; Satoshi Shuto; Mitsuhiro Arisawa

Publisher: John Wiley and Sons
Year: 2009
Tongue: English
Weight: 194 KB
Volume: 2009
Category: Article
ISSN: 1434-193X
DOI: 10.1002/ejoc.200900520

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✦ Synopsis

Abstract

A steric and electronic effect on enamide/ene metathesis, a novel preparation of 2‐substituted indoles and 3‐substituted indoles using enamide‐ene metathesis as a key reaction, and its application to the synthesis of indomethacin are described. (© Wiley‐VCH Verlag GmbH & Co. KGaA, 69451 Weinheim, Germany, 2009)

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