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An in-vitro cocktail assay for assessing compound-mediated inhibition of six major cytochrome P450 enzymes

✍ Scribed by Wang, Jing-Jing; Guo, Jian-Jun; Zhan, Jenny; Bu, Hai-Zhi; Lin, Jiunn H.


Book ID
121647029
Publisher
Elsevier
Year
2014
Tongue
English
Weight
999 KB
Volume
4
Category
Article
ISSN
2095-1779

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In vitro interaction cocktail assay for
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## Abstract A sensitive and rugged LC/MSMS method was developed for a comprehensive __in vitro__ metabolic interaction screening assay with N‐in‐1 approach reported earlier. A cocktail consisting of ten cytochrome P450 (CYP)‐selective probe substrates with known kinetic, metabolic and interaction p