Difficulties encountered in the synthesis of resin-bound secondary amines attached via an acid-labile linker encouraged us to employ an alternative approach. A one-pot, scalable procedure for the synthesis of Fmoc-protected, amine/linker constructs is reported. These compounds can be efficiently cou
An improved two-resin method for the cleavage of tertiary amines from REM resin
✍ Scribed by Carolina Alhambra; Julia Castro; Jose Luis Chiara; Esther Fernández; Alfonso Fernández-Mayoralas; José M Fiandor; Silvestre Garcı́a-Ochoa; Marı́a D Martı́n-Ortega
- Publisher
- Elsevier Science
- Year
- 2001
- Tongue
- French
- Weight
- 139 KB
- Volume
- 42
- Category
- Article
- ISSN
- 0040-4039
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