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An amidyl radical cyclisation approach towards the synthesis of β-lactams

✍ Scribed by Andrew J. Clark; Joanne L. Peacock

Publisher
Elsevier Science
Year
1998
Tongue
French
Weight
200 KB
Volume
39
Category
Article
ISSN
0040-4039

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✦ Synopsis

Amidyl radicals generated from tributylstannane mediated homolysis of O-benzoyl hydroxamic acid derivatives (2a,d) underl~o 4-exo trig cyclisation to furnish 13-1actam derivatives (4ad).

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