## Abstract Structure‐based quantitative structure‐activity relationship (QSAR) studies on a series of checkpoint kinase 1 (Chk1) inhibitors were performed to find the key structural features responsible for their inhibitory activity. Molecular docking was employed to explore the binding mode of al
Aminopyridinecarboxamide-based inhibitors: Structure–activity relationship
✍ Scribed by Dominique F. Bonafoux; Sheri L. Bonar; Michael Clare; Ann M. Donnelly; Jeanette L. Glaenzer; Julia A. Guzova; He Huang; Nandidni N. Kishore; Francis J. Koszyk; Patrick J. Lennon; Adam Libby; Sumathy Mathialagan; David S. Oburn; Sharon A Rouw; Cynthia D. Sommers; Catherine S. Tripp; Lori J. Vanella; Richard Weier; Serge G. Wolfson; Horng-Chih Huang
- Book ID
- 108072745
- Publisher
- Elsevier Science
- Year
- 2010
- Tongue
- English
- Weight
- 823 KB
- Volume
- 18
- Category
- Article
- ISSN
- 0968-0896
No coin nor oath required. For personal study only.
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