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Aminocyanopyridine inhibitors of mitogen activated protein kinase-activated protein kinase 2 (MK-2)

✍ Scribed by David R. Anderson; Shridhar Hegde; Emily Reinhard; Leslie Gomez; William F. Vernier; Len Lee; Shuang Liu; Aruna Sambandam; Patricia A. Snider; Liaqat Masih


Book ID
108073569
Publisher
Elsevier Science
Year
2005
Tongue
English
Weight
120 KB
Volume
15
Category
Article
ISSN
0960-894X

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A class of inhibitors of mitogen activated protein kinase-activated kinase 2 (MK2) was discovered via high-throughput screening. This compound class demonstrates activity against the enzyme with sub-microM IC(50) values, and suppresses LPS-induced TNFalpha levels in THP-1 cells. MK2 inhibition kinet