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Acid-catalyzed rearrangement of 3-(β-2-aminostyryl)quinoxalin-2(1H)ones—a new and efficient method for the synthesis of 2-benzimidazol-2-ylquinolines

✍ Scribed by Vakhid A. Mamedov; Dina F. Saifina; Aidar T. Gubaidullin; Venera R. Ganieva; Saniya F. Kadyrova; Dimitry V. Rakov; Il’dar Kh. Rizvanov; Oleg G. Sinyashin


Publisher
Elsevier Science
Year
2010
Tongue
French
Weight
316 KB
Volume
51
Category
Article
ISSN
0040-4039

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✦ Synopsis


1

H NMR data X-ray diffraction analysis a b s t r a c t A highly efficient, one-step, versatile method for the synthesis of 2-benzimidazol-2-ylquinolines has been developed on the basis of an acid-catalyzed rearrangement proceeding via a novel ring contraction of 3-(b-2-aminostyryl)quinoxalin-2(1H)ones.


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