A versatile synthesis of 4-aryl tetrahyd
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Paul R Eastwood
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Article
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2000
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Elsevier Science
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French
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A simple preparation of cyclic vinyl boronates derived from the vinyl triflates of N-protected tetrahydropyridines is described. Suzuki coupling of the boronates with aryl bromides, iodides and triflates proceeds in good yield to give 4-aryl tetrahydropyridines.