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A versatile new synthesis of 4-aryl- and heteroaryl-[3,4-c]pyrrolocarbazoles by [4+2] cycloaddition followed by palladium catalysed cross coupling

โœ Scribed by Gary McCort; Olivier Duclos; Caroline Cadilhac; Eric Guilpain

Publisher
Elsevier Science
Year
1999
Tongue
French
Weight
242 KB
Volume
40
Category
Article
ISSN
0040-4039

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โœฆ Synopsis

4-Bromo-and 4-trifluorosulfonyloxypyrrolo[3,4-c]carbazoles were prepared in five steps via a [4+2] cycloaddition and were used as key intermediates in paUadium-catalysed cross coupling reactions allowing the rapid generation of structurally diverse protein kinase C inhibitors.

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