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A useful method for the preparation of fully protected peptide acids and esters

✍ Scribed by André Pichette; Normand Voyer; Rémi Larouche; Jean-Christophe Meillon

Publisher
Elsevier Science
Year
1997
Tongue
French
Weight
175 KB
Volume
38
Category
Article
ISSN
0040-4039

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✦ Synopsis

Resin bound peptides can be cleaved from the Kaiser oxime resin using various oxygen nucleophiles (H20, CH3OH, PhCH2OH) with DBU. Fully protected peptide acids and esters are obtained rapidly and with good yields using this new method of cleavage.

📜 SIMILAR VOLUMES

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A practical method for the preparation of protected peptide fragments using the Kaiser oxime resin
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