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A stereo-divergent route to aminocyclopentitol derivatives

✍ Scribed by Shital K. Chattopadhyay; Ayan Bandyopadhyay

Book ID
104099334
Publisher
Elsevier Science
Year
2011
Tongue
French
Weight
372 KB
Volume
52
Category
Article
ISSN
0040-4039

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✦ Synopsis

A stereo-divergent synthetic strategy based on diastereoselective vinylation of an a-amino aldehyde, ring-closing metathesis reaction and diastereoselective dihydroxylation reaction as key steps has been developed for the synthesis of three aminocyclopentitol derivatives of chemical and biological relevance.

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