๐”– Bobbio Scriptorium
โœฆ   LIBER   โœฆ

A simple strategy for the synthesis of hydroxyethylene dipeptide isostere from D-glucose

โœ Scribed by T.K. Chakraborty; K. Azhar Hussain; D. Thippeswamy


Publisher
Elsevier Science
Year
1995
Tongue
French
Weight
557 KB
Volume
51
Category
Article
ISSN
0040-4020

No coin nor oath required. For personal study only.


๐Ÿ“œ SIMILAR VOLUMES


Diastereoselective synthesis of the key
โœ Bharat R. Lagu; Dennis C. Liotta ๐Ÿ“‚ Article ๐Ÿ“… 1994 ๐Ÿ› Elsevier Science ๐ŸŒ French โš– 313 KB

Abatraot: An efficient and hiihly stereoselective route for preparing hydroxyethylene dipeptide isosteres from a-N,Ndibenzylamino ketones has been developed. In the last few years hydroxyethylene dipeptide isosteres ("peptide mimics') have generated considerable interest in the scientific community

New synthesis of 5-amino-4-hydroxy-2,6-d
โœ Fabio Benedetti; Paolo Maman; Stefano Norbedo ๐Ÿ“‚ Article ๐Ÿ“… 2000 ๐Ÿ› Elsevier Science ๐ŸŒ French โš– 73 KB

Two stereoisomers of the title compound have been synthesized from the methyl ester of N-Boc L-valine. The aminoester was initially converted into an a%-amino a,b-unsaturated ketone via a phosphonoketone and a Horner-Emmons olefination with acetaldehyde. Hydrocyanation of the enone with diethylalumi

Amino-alcohol dipeptide analogues: A sim
โœ R.J. Arrowsmith; D.E Davies; Y.C. Fogden; C.J. Harris; C. Thompson ๐Ÿ“‚ Article ๐Ÿ“… 1987 ๐Ÿ› Elsevier Science ๐ŸŒ French โš– 155 KB

Two sample approaches to an ammo-alcohol isostere of proteolytrcally-cleavable dipeptrde sequences are descrrbed; this isostere is incorporated into stereochemically-defined tetrapeptlde analogues. We1 and others2 have shown that replacement of the cleavable amrde bond of appropriate peptide substra