✦ LIBER ✦

A short synthesis of 3(r)-hydroxy-2(R)-isopropyltetrahydrothiophene: A precursor to a high-affinity P2-ligand of HIV-1 protease inhibitors

✍ Scribed by B.Moon Kim; Hee-Yoon Lee; Peter M. Munson; James P. Guare; Colleen McDonough

Publisher: Elsevier Science
Year: 1993
Tongue: French
Weight: 302 KB
Volume: 34
Category: Article
ISSN: 0040-4039
DOI: 10.1016/0040-4039(93)88093-x

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

ChemInform Abstract: A Facile Synthesis

ChemInform Abstract: A Facile Synthesis of (2R,3S)-1-Amino-3-tert-butoxycarbonylamino-2-hydroxy-4-phenylbutane: A Useful Component Block of HIV Protease Inhibitor.

✍ YOKO YUASA; YOSHIFUMI YUASA; H. TSURUTA 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 34 KB 👁 1 views

ChemInform Abstract: A Practical Synthes

ChemInform Abstract: A Practical Synthesis of (1S,2R)-1-Amino-2-indanol, a Key Component of HIV Protease Inhibitor, Indinavir.

✍ H. KAJIRO; S. MITAMURA; A. MORI; T. HIYAMA 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 35 KB 👁 2 views

Corrigendum to “Enantioselective synthes

Corrigendum to “Enantioselective synthesis of cyclopentyltetrahydrofuran (Cp-THF), an important high-affinity P2-ligand for HIV-1 protease inhibitors”: [Tetrahedron Lett. 49 (2008) 3409]

✍ Arun K. Ghosh; Jun Takayama 📂 Article 📅 2008 🏛 Elsevier Science 🌐 French ⚖ 114 KB

ChemInform Abstract: A Practical Synthes

ChemInform Abstract: A Practical Synthesis of (1S,2R)-1-Amino-2-indanol, a Key Component of an HIV Protease Inhibitor, Indinavir.

✍ Hiroshi Kajiro; Shuichi Mitamura; Atsunori Mori; Tamejiro Hiyama 📂 Article 📅 2010 🏛 John Wiley and Sons ⚖ 30 KB 👁 2 views

An expeditious synthesis of (2R,3S)-3-te

An expeditious synthesis of (2R,3S)-3-tert-butoxycarbonylamino-1-isobutylamino-4-phenyl-2-butanol, a key building block of HIV protease inhibitors

✍ Norio Shibata; Tadashi Katoh; Shiro Terashima 📂 Article 📅 1997 🏛 Elsevier Science 🌐 French ⚖ 134 KB

A Convenient Synthesis of the Echinacea-

A Convenient Synthesis of the Echinacea-Derived Immunostimulator and HIV-1 Integrase Inhibitor (−)-(2R,3R)-Chicoric Acid

✍ Anne-Marie Lamidey; Lionel Fernon; Laurent Pouységu; Charlotte Delattre; Stéphan 📂 Article 📅 2002 🏛 John Wiley and Sons 🌐 German ⚖ 87 KB 👁 2 views

The Echinacea-derived immunostimulator and HIV-1 integrase inhibitor (À)-chicoric acid ( 2,3-bis{[3-(3,4-dihydroxyphenyl)-1-oxoprop-2-enyl]oxy}butanedioic acid; 1a) was conveniently prepared via a silanepromoted Pd-mediated chemoselective hydrogenolysis of its perbenzylated derivative 12a, which was