✦ LIBER ✦

A QSAR Approach to the Study of Structural Requirements of Muscarinic Receptor Ligands Part II: Antagonists

✍ Scribed by Pratesi, P. ;Caliendo, G. ;Silipo, C. ;Vittoria, A.

Book ID: 112185389
Publisher: John Wiley and Sons
Year: 1992
Tongue: English
Weight: 950 KB
Volume: 11
Category: Article
ISSN: 1611-020X
DOI: 10.1002/qsar.19920110205

No coin nor oath required. For personal study only.

📜 SIMILAR VOLUMES

Chemometric approach to a QSAR study of

Chemometric approach to a QSAR study of peptides behaving as NK-2 receptor antagonists

✍ Sergio Clementi; Gabriele Cruciani; Daniela Riganelli; Paolo Rovero; Vittorio Pe 📂 Article 📅 1990 🏛 Elsevier Science ⚖ 578 KB

This paper shows the advantages of using chemometric strategies in QSAR of NKA analogues containing D-Tryptophan and behaving as highly selective NK-2 receptor antagonists: a) detecting the sequence with optimal antagonist activity, and b) having a strategy for selecting a few most informative seque

A 3D QSAR approach to the search for geo

A 3D QSAR approach to the search for geometrical similarity in a series of nonpeptide angiotensin II receptor antagonists

✍ Laura Belvisi; Gianpaolo Bravi; Carlo Scolastico; Anna Vulpetti; Aldo Salimbeni; 📂 Article 📅 1994 🏛 Springer Netherlands 🌐 English ⚖ 721 KB

A 3D QSAR methodology based on the combined use of conformational analysis and chemometrics was applied to perform a comparative analysis of the 3D conformational features of 13 nonpeptide angiotensin II receptor antagonists showing different levels of binding affinity. Conformational analysis by us

Tandem 3D-QSARs Approach as a Valuable T

Tandem 3D-QSARs Approach as a Valuable Tool to Predict Binding Affinity Data: Design of New Gly/NMDA Receptor Antagonists as a Key Study.

✍ S. Moro; et al. et al. 📂 Article 📅 2007 🏛 John Wiley and Sons ⚖ 11 KB 👁 1 views

Tandem 3D-QSARs Approach as a Valuable T

Tandem 3D-QSARs Approach as a Valuable Tool To Predict Binding Affinity Data: Design of New Gly/NMDA Receptor Antagonists as a Key Study

✍ Bacilieri, M.; Varano, F.; Deflorian, F.; Marini, M.; Catarzi, D.; Colotta, V.; 📂 Article 📅 2007 🏛 American Chemical Society 🌐 English ⚖ 419 KB

Probing the Pharmacophore for Allosteric

Probing the Pharmacophore for Allosteric Ligands of Muscarinic M 2 Receptors: SAR and QSAR Studies in a Series of Bisquaternary Salts of Caracurine V and Related Ring Systems

✍ Zlotos, Darius P.; Buller, Stefan; Stiefl, Nikolaus; Baumann, Knut; Mohr, Klaus 📂 Article 📅 2004 🏛 American Chemical Society 🌐 English ⚖ 278 KB

Insight into the structural requirement

Insight into the structural requirement of aryltriazolinone derivatives as angiotensin II AT1receptor: 2D and 3D-QSAR k-Nearest Neighbor Molecular Field Analysis approach

✍ Mukesh C. Sharma, D. V. Kohli 📂 Article 📅 2011 🏛 Springer-Verlag 🌐 English ⚖ 701 KB