A series of 2-alkyl and 2-cycioalkyl raloxifene analogs have been prepared and evaluated in both in vitro and in vivo models of estrogen/antiestrogen activity. In particular, the 2-cyclohexyl analogs show promise as potent sdective estrogen-receptor modulators (SERMs). The decreased production of o
A pharmacological review of raloxifene
โ Scribed by Henry U. Bryant; Andrew L. Glasebrook; Na N. Yang; Masahiko Sato
- Publisher
- Springer
- Year
- 1996
- Tongue
- English
- Weight
- 951 KB
- Volume
- 14
- Category
- Article
- ISSN
- 0914-8779
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