A novel solid-phase chlorinating reagent for the synthesis of acyl chlorides
β Scribed by Guanglin Luo; Li Xu; Graham S. Poindexter
- Publisher
- Elsevier Science
- Year
- 2002
- Tongue
- French
- Weight
- 199 KB
- Volume
- 43
- Category
- Article
- ISSN
- 0040-4039
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π SIMILAR VOLUMES
A novel, mild method for the synthesis of di-and trisubstituted N-acyl ureas on solid support is described. Addition of carboxylic acids to a resin-bound carbimidoyl chloride gave, initially, an O-acyl isourea which subsequently rearranged to the corresponding N-acyl urea. Trisubstituted N-acyl urea
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